European Journal of Pharmacology: Molecular Pharmacology
Volume 290, Issue 1, 23 June 1995, Pages 29-36
Pramipexole binding and activation of cloned and expressed dopamine D2, D3 and D4 receptors
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2021, Pharmacological ResearchCitation Excerpt :PPX also has affinity for D4R [50], but the evidence that D4R is not expressed in the nigrostriatal system [12] rules out its participation in this phenomenon. It should be noted that although PPX has a higher affinity for D3R than for D2R, its Kd for D2R is not more than 5–7 fold higher than for D3R [50,51]. Furthermore, D2R expression in the mesostriatal system is about one order of magnitude higher than that of D3R [52].
Copyright © 1995 Published by Elsevier B.V.